Molecule Details
InChIKeyXNUXIYGMZDJLFB-UHFFFAOYSA-N
Compound Name3-(1-Cyclopropylcyclopropyl)-8-(cyclopropylmethyl)-2,4,5,8,13-pentazatricyclo[7.4.0.02,6]trideca-1(9),3,5,10-tetraene-7,12-dione
Canonical SMILESO=c1c2nnc(C3(C4CC4)CC3)n2c2nc(O)ccc2n1CC1CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q14123 PDE1C Homo sapiens Human PF00233 PF08499 8.6 IC50 ChEMBL;BindingDB
P54750 PDE1A Homo sapiens Human PF00233 PF08499 8.6 IC50 ChEMBL;BindingDB
Q01064 PDE1B Homo sapiens Human PF00233 PF08499 8.5 IC50 ChEMBL;BindingDB