Molecule Details
InChIKeyXNRMQSNQFCESPA-UHFFFAOYSA-N
Compound Name3-(2,4-dimethylbenzoyl)-1-(4-fluorobenzoyl)-1H-pyrazole
Canonical SMILESCc1ccc(C(=O)c2ccn(C(=O)c3ccc(F)cc3)n2)c(C)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.15
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08246 ELANE Homo sapiens Human PF00089 7.6 Ki ChEMBL;BindingDB
P00734 F2 Homo sapiens Human PF00594 PF00051 PF09396 PF00089 6.9 IC50 ChEMBL;BindingDB
Q99895 CTRC Homo sapiens Human PF00089 6.9 IC50 BindingDB