Target not found.
Molecule Details
InChIKeyXNEWLEJBYAVWCK-UHFFFAOYSA-N
Compound Name2-(3,4-dichlorophenyl)-N-(4-fluoro-3-trifluoromethylbenzyl)-2,N-dimethyl-4-[4-(2-oxo-pyrrolidin-1-yl)-piperidin-1-yl]-butyramide
Canonical SMILESCN(Cc1ccc(F)c(C(F)(F)F)c1)C(=O)C(C)(CCN1CCC(N2CCCC2=O)CC1)c1ccc(Cl)c(Cl)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.6
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29371 TACR3 Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P21452 TACR2 Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB
P25103 TACR1 Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB