Molecule Details
InChIKeyXMTCSFQKNADGEY-UHFFFAOYSA-O
Compound Name2-[[(3-amino-6-chloropyrazine-2-carbonyl)amino]methyl]-N-[2-(dimethylamino)ethyl]-1,3-diethyl-N-methylbenzimidazol-1-ium-5-carboxamide
Canonical SMILESCCn1c(CNC(=O)c2nc(Cl)cnc2N)[n+](CC)c2ccc(C(=O)N(C)CCN(C)C)cc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.77
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P37088 SCNN1A Homo sapiens Human PF00858 7.8 IC50 ChEMBL
P51168 SCNN1B Homo sapiens Human PF00858 7.8 IC50 ChEMBL
P51170 SCNN1G Homo sapiens Human PF00858 7.8 IC50 ChEMBL