Molecule Details
InChIKeyXLXSAKCOAKORKW-YBKDWAIYSA-N
Compound NameH-DL-Pyr-His-Trp-Ser-Tyr-Gly-Leu-Arg-D-Pro-Gly-NH2
Canonical SMILESCC(C)C[C@H](NC(=O)CNC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)C1CCC(=O)N1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1CCC[C@@H]1C(=O)NCC(N)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.75
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P41145 OPRK1 Homo sapiens Human PF00001 10.4 Ki ChEMBL
P41146 OPRL1 Homo sapiens Human PF00001 7.1 Ki ChEMBL