Molecule Details
InChIKeyXLWHWNHGNRPPBH-JOCHJYFZSA-N
Compound Name(2R)-2-[[2-(1H-indole-2-carbonylamino)benzoyl]amino]-4-phenylbutanoic acid
Canonical SMILESO=C(Nc1ccccc1C(=O)N[C@H](CCc1ccccc1)C(=O)O)c1cc2ccccc2[nH]1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.15
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 8.3 Ki ChEMBL;BindingDB
P32239 CCKBR Homo sapiens Human PF00001 6.0 Ki ChEMBL;BindingDB