Molecule Details
InChIKeyXLAHTLJMVQSDTK-PQQNNWGCSA-N
Compound Name(10S,13R)-13-(benzylsulfonylamino)-N-[(4-carbamimidoylphenyl)methyl]-3,12,20-trioxo-1,4,11,19,22-pentazatetracyclo[20.3.2.25,8.215,18]hentriaconta-5,7,15(29),16,18(28),30-hexaene-10-carboxamide
Canonical SMILESN=C(N)c1ccc(CNC(=O)[C@@H]2Cc3ccc(cc3)NC(=O)CN3CCCN(CC3)CC(=O)Nc3ccc(cc3)C[C@@H](NS(=O)(=O)Cc3ccccc3)C(=O)N2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.83
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P00747 PLG Homo sapiens Human PF00051 PF00024 PF00089 9.2 Ki ChEMBL;BindingDB
P03952 KLKB1 Homo sapiens Human PF00024 PF00089 6.4 Ki ChEMBL;BindingDB