Molecule Details
InChIKeyXKEPASMYHMOCPP-UHFFFAOYSA-N
Compound Name2-[3-(Tert-butylamino)-6-fluoro-2-methylquinoxalin-5-yl]-1,5-dihydropyrrolo[3,2-c]pyridin-4-one
Canonical SMILESCc1nc2ccc(F)c(-c3cc4c(=O)[nH]ccc4[nH]3)c2nc1NC(C)(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.81
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9P1W9 PIM2 Homo sapiens Human PF00069 10.0 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 9.6 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 6.8 IC50 ChEMBL