Molecule Details
InChIKeyXKDSMPCDGPJCLX-UHFFFAOYSA-N
Canonical SMILESc1ccc(-c2nnc(-c3ccc4[nH]cc(-c5cncc(C6CC6)n5)c4c3)o2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.81
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB