Molecule Details
InChIKeyXJRUWGFZGQNPPD-UHFFFAOYSA-N
Compound Name6-but-3-enyl-4-[1-methyl-6-(morpholine-4-carbonyl)benzimidazol-4-yl]-1H-pyrrolo[2,3-c]pyridin-7-one
Canonical SMILESC=CCCn1cc(-c2cc(C(=O)N3CCOCC3)cc3c2ncn3C)c2cc[nH]c2c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.24
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15544 TAF11 Homo sapiens Human PF04719 9.0 Kd ChEMBL;BindingDB
Q8IZX4 TAF1L Homo sapiens Human PF00439 PF12157 PF09247 PF15288 8.3 Kd ChEMBL;BindingDB
P21675 TAF1 Homo sapiens Human PF00439 PF12157 PF09247 PF15288 7.4 IC50 ChEMBL;BindingDB