Molecule Details
InChIKeyXJPIRGSNEBMRTI-KXQOOQHDSA-N
Compound NameCID 87332775
Canonical SMILESCC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(N[C@H](CCN5CCOCC5)CSc5ccccc5)c(S(=O)(=O)C(F)(F)Cl)c4)cc3)CC2)=C(c2ccc(Cl)cc2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.45
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P10415 BCL2 Homo sapiens Human PF00452 PF02180 10.3 Ki ChEMBL
Q07817 BCL2L1 Homo sapiens Human PF00452 PF02180 9.3 Ki ChEMBL
Q92843 BCL2L2 Homo sapiens Human PF00452 PF02180 8.7 Ki ChEMBL