Molecule Details
InChIKeyXJIWJTAALOWWFJ-RASJINCSSA-N
Compound NameN-[(S)-1-(2-{4-[(3R,4S)-4-(4-Chloro-phenyl)-1-(tetrahydro-pyran-4-YL)-pyrrolidine-3-carbonyl]-piperazin-1-YL}-5-methyl-phenyl)-2-methyl-propyl]-3-dimethylamino-propionamide
Canonical SMILESCc1ccc(N2CCN(C(=O)[C@H]3CN(C4CCOCC4)C[C@@H]3c3ccc(Cl)cc3)CC2)c([C@@H](NC(=O)CCN(C)C)C(C)C)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.99
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32245 MC4R Homo sapiens Human PF00001 7.8 IC50 ChEMBL;BindingDB
Q01726 MC1R Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB
P33032 MC5R Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB