Molecule Details
InChIKeyXIXCDPUONOFFOT-UHFFFAOYSA-N
Compound Name4-(1-Isopropyl-2-methylimidazol-5-yl)-2-[4-(3-morpholinopropylsulphonyl)anilino]pyrimidine
Canonical SMILESCc1ncc(-c2ccnc(Nc3ccc([S@SP3](=O)(=O)CCCN4CCOCC4)cc3)n2)n1C(C)C
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.48
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.5 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 7.5 pIC50 TTD_MultiTarget