Molecule Details
InChIKeyXIVVAPJAZVPZQR-HSZRJFAPSA-N
Compound NameN-[(3R)-6-cyano-1-[(3-methylimidazol-4-yl)methyl]-3,4-dihydro-2H-quinolin-3-yl]-N-(thiophen-3-ylmethyl)benzenesulfonamide
Canonical SMILESCn1cncc1CN1C[C@H](N(Cc2ccsc2)S(=O)(=O)c2ccccc2)Cc2cc(C#N)ccc21
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.55
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.6 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.6 IC50 ChEMBL