Molecule Details
InChIKeyXIJOBJBWOPBBNG-UHFFFAOYSA-N
Compound Name6-methyl-2-(3-methyl-5-((4-methylphenyl)amino)-1H-pyrazol-1-yl)-1,4-dihydropyrimidin-4-one
Canonical SMILESCc1ccc(Nc2cc(C)nn2-c2nc(C)cc(O)n2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.34
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O95977 S1PR4 Homo sapiens Human PF00001 6.8 IC50 ChEMBL
P41145 OPRK1 Homo sapiens Human PF00001 6.1 IC50 ChEMBL;BindingDB
P21453 S1PR1 Homo sapiens Human PF00001 6.1 IC50 ChEMBL