Molecule Details
InChIKeyXIICSQSWOYKKRN-VPUSJEBWSA-N
Compound Name2-[4-[[(2R)-2-[[(2S)-3-(3-bromophenyl)-2-[(4-phenylbenzoyl)amino]propanoyl]amino]-2-cyanoethoxy]methyl]triazol-1-yl]acetic acid
Canonical SMILESN#C[C@H](COCc1cn(CC(=O)O)nn1)NC(=O)[C@H](Cc1cccc(Br)c1)NC(=O)c1ccc(-c2ccccc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.83
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P07858 CTSB Homo sapiens Human PF00112 PF08127 7.6 Ki ChEMBL;BindingDB
P43235 CTSK Homo sapiens Human PF08246 PF00112 6.5 Ki ChEMBL;BindingDB
P25774 CTSS Homo sapiens Human PF08246 PF00112 6.5 Ki ChEMBL;BindingDB