Molecule Details
InChIKeyXIELCZGHLSBOSH-UHFFFAOYSA-N
Compound Name4-[9-[3-[(4-methoxyphenyl)sulfonylamino]phenyl]-3,3,6,6-tetramethyl-1,8-dioxo-4,5,7,9-tetrahydro-2H-acridin-10-yl]benzenesulfonamide
Canonical SMILESCOc1ccc(S(=O)(=O)Nc2cccc(C3C4=C(CC(C)(C)CC4=O)N(c4ccc(S(N)(=O)=O)cc4)C4=C3C(=O)CC(C)(C)C4)c2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 6.6 Ki ChEMBL;BindingDB
Q16790 CA9 Homo sapiens Human PF00194 6.1 Ki ChEMBL;BindingDB
O43570 CA12 Homo sapiens Human PF00194 6.0 Ki ChEMBL;BindingDB