Molecule Details
InChIKeyXGLOKDGUVCNLTH-UHFFFAOYSA-N
Compound NameN-(4-sulfamoylphenyl)-4-[3,3,6,6-tetramethyl-1,8-dioxo-9-[3-[3,3,6,6-tetramethyl-1,8-dioxo-10-[4-[(4-sulfamoylphenyl)carbamoyl]phenyl]-4,5,7,9-tetrahydro-2H-acridin-9-yl]phenyl]-4,5,7,9-tetrahydro-2H-acridin-10-yl]benzamide
Canonical SMILESCC1(C)CC(=O)C2=C(C1)N(c1ccc(C(=O)Nc3ccc(S(N)(=O)=O)cc3)cc1)C1=C(C(=O)CC(C)(C)C1)C2c1cccc(C2C3=C(CC(C)(C)CC3=O)N(c3ccc(C(=O)Nc4ccc(S(N)(=O)=O)cc4)cc3)C3=C2C(=O)CC(C)(C)C3)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.98
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 7.5 Ki ChEMBL;BindingDB
P43166 CA7 Homo sapiens Human PF00194 7.3 Ki ChEMBL;BindingDB
P00915 CA1 Homo sapiens Human PF00194 6.1 Ki ChEMBL;BindingDB