Molecule Details
InChIKeyXGDNBPSADFJVLS-UHFFFAOYSA-N
Compound Name4,5-Dichloro-6-[({[(4-methylphenyl)sulfonyl]amino}carbonyl)amino]benzene-1,3-disulfonamide
Canonical SMILESCc1ccc(S(=O)(=O)NC(=O)Nc2c(S(N)(=O)=O)cc(S(N)(=O)=O)c(Cl)c2Cl)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.98
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00915 CA1 Homo sapiens Human PF00194 8.1 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 7.9 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.9 pIC50 TTD_MultiTarget