Molecule Details
InChIKeyXECCFMIBBHXKBJ-UHFFFAOYSA-N
Compound Name7-(4-fluoro-1H-pyrazol-1-yl)-2-((3-fluoropyridin-2-yl)methyl)-8-(3-methylimidazo[l,2-a]pyridin-6-yl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-amine
Canonical SMILESCc1cnc2ccc(-c3c(-n4cc(F)cn4)nc(N)n4nc(Cc5ncccc5F)nc34)cn12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.5
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29274 ADORA2A Homo sapiens Human PF00001 9.7 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 8.0 IC50 ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 7.8 IC50 ChEMBL;BindingDB