Molecule Details
InChIKeyXDRQTCJBCDWMJW-UHFFFAOYSA-N
Compound Name6-(2-aminoethylsulfonyl)-3-(2-amino-7-methyl-3H-benzimidazol-4-yl)-2-(2H-tetrazol-5-yl)benzenesulfonamide
Canonical SMILESCc1ccc(-c2ccc(S(=O)(=O)CCN)c(S(N)(=O)=O)c2-c2nn[nH]n2)c2nc(N)[nH]c12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.79
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 10.0 IC50 BindingDB
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.9 IC50 ChEMBL;BindingDB
P52699 Serratia marcescens Pathogen PF00753 9.4 IC50 BindingDB