Molecule Details
InChIKeyXDNNQWBDYFHHSY-UHFFFAOYSA-N
Compound NamePHA-927F free base
Canonical SMILESCC(C)Nc1nc(Cl)c(-c2cc(N)cc(C(=O)O)c2)n(CC(=O)NCc2ccc(C(=N)N)cc2)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.6
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08709 F7 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 7.8 IC50 ChEMBL;BindingDB
P13726 F3 Homo sapiens Human PF09294 PF01108 7.8 IC50 ChEMBL
P07477 PRSS1 Homo sapiens Human PF00089 7.2 IC50 ChEMBL;BindingDB