Molecule Details
InChIKeyXDGHTBHPIPZHLJ-UHFFFAOYSA-N
Compound NameN-methyl-6-(2-methyl-5-(5-(trifluoromethyl)-1Hbenzo[d]imidazol-2-ylamino)phenyl)quinazolin-2-amine
Canonical SMILESCNc1ncc2cc(-c3cc(Nc4nc5cc(C(F)(F)F)ccc5[nH]4)ccc3C)ccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16539 MAPK14 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB
P06239 LCK Homo sapiens Human PF07714 PF00017 PF00018 6.5 IC50 ChEMBL;BindingDB