Molecule Details
InChIKeyXCUISAPLRLETKW-UHFFFAOYSA-N
Compound Namen-[6-(2-Furyl)-5-pyridin-4-ylpyrazin-2-yl]cyclobutanecarboxamide
Canonical SMILESO=C(Nc1cnc(-c2ccncc2)c(-c2ccco2)n1)C1CCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.71
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29275 ADORA2B Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB