Molecule Details
InChIKeyXCQPCESBLWIBEC-UHFFFAOYSA-N
Compound NameN-[3-[4-(3-chloro-2-methylphenyl)piperazin-1-yl]propyl]-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-2,5-dimethylimidazole-4-carboxamide
Canonical SMILESCc1c(Cl)cccc1N1CCN(CCCNC(=O)c2nc(C)n(-c3ccc4c(c3)OCCO4)c2C)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 8.6 IC50 ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 7.5 IC50 ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 7.0 IC50 ChEMBL;BindingDB