Molecule Details
InChIKeyXBLGRIMBLMBXMW-UHFFFAOYSA-N
Compound NameN-(1-Benzylpiperidin-4-yl)-4-(2,6-dioxo-1-propyl-2,3,6,7-tetrahydro-1H-purin-8-yl)benzenesulfonamide
Canonical SMILESCCCn1c(=O)[nH]c2nc(-c3ccc(S(=O)(=O)NC4CCN(Cc5ccccc5)CC4)cc3)[nH]c2c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.77
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P29275 ADORA2B Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB