Molecule Details
InChIKeyXBFRRCZSSOFGAI-UHFFFAOYSA-N
Compound NameN-[4-[2-ethyl-5-(4-fluorophenyl)-1H-imidazol-4-yl]-2-pyridinyl]cyclopropanecarboxamide
Canonical SMILESCCc1nc(-c2ccc(F)cc2)c(-c2ccnc(NC(=O)C3CC3)c2)[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.09
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16539 MAPK14 Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
P49841 GSK3B Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB
P49840 GSK3A Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB