Molecule Details
InChIKeyWZPMLZHTAAYDCQ-UHFFFAOYSA-N
Compound Name2-{[7-Acetyl-3-(2-furylmethyl)-4-oxo-3,4,5,6,7,8-hexahydropyrido[4',3':4,5]thieno[2,3-D]pyrimidin-2-YL]sulfanyl}-N-(5-chloro-2-methylphenyl)acetamide
Canonical SMILESCC(=O)N1CCc2c(sc3nc(SCC(=O)Nc4cc(Cl)ccc4C)n(Cc4ccco4)c(=O)c23)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.59
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P25440 BRD2 Homo sapiens Human PF17035 PF00439 6.9 IC50 ChEMBL;BindingDB
Q15059 BRD3 Homo sapiens Human PF17035 PF00439 6.8 IC50 ChEMBL;BindingDB
O60885 BRD4 Homo sapiens Human PF17035 PF17105 PF00439 6.1 IC50 ChEMBL;BindingDB