InChIKey	WZDGZWOAQTVYBX-XOINTXKNSA-N
Compound Name	Tibolone
Canonical SMILES	C#C[C@]1(O)CC[C@H]2[C@@H]3[C@H](C)CC4=C(CCC(=O)C4)[C@H]3CC[C@@]21C
Clinical Status	Data-mined Candidate
Targets (Human+Pathogen)	2
Pfam Stratification	Cross-Family
Avg pChEMBL	6.91
Source	ChEMBL

DrugBank ID	DB09070
Drug Name	Tibolone
CAS Number	5630-53-5
Groups	approved investigational
ATC Codes	G03CX01
Description	Tibolone is a synthetic steroid hormone drug, which is mainly non-selective in its binding profile, acting as an agonist primarily at estrogen receptors (ER), with a preference for ER alpha [L1874]. Tibolone (Livial, Org OD 14), produced by Organon (West Orange, NJ), is a synthetic steroid that poss...

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Categories: Anabolic Agents Antineoplastic Agents, Hormonal Cardiovascular Agents Estrogen Receptor Modulators Estrogens Estrogens, Antiestrogens, and Estrogen Agonist-Antagonists Fused-Ring Compounds Genito Urinary System and Sex Hormones Hormone Antagonists Hormones Hormones, Hormone Substitutes, and Hormone Antagonists Norpregnanes Norsteroids Sex Hormones and Modulators of the Genital System Steroids

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Cross-references: ChEBI: 32223 CHEMBL2103774 ChemSpider: 392038 Drugs Product Database (DPD): 1251 D01639 PubChem:444008 PubChem:347827821 RxCUI: 38260 Wikipedia: Tibolone ZINC: ZINC000003812889