Molecule Details
InChIKeyWYLBWIZCNKSPCW-SFHVURJKSA-N
Compound Name4''-{1-[(2S)-pyrrolidin-2-ylmethyl]piperidin-4-yl}-2-(1H-tetrazol-5-yl)-4-(trifluoromethyl)biphenyl-3-sulfonamide
Canonical SMILESNS(=O)(=O)c1c(C(F)(F)F)ccc(-c2ccc(C3CCN(C[C@@H]4CCCN4)CC3)cc2)c1-c1nnn[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.54
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P52699 Serratia marcescens Pathogen PF00753 9.2 IC50 BindingDB
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 8.4 IC50 ChEMBL;BindingDB
Q5GN09 vim-1 Klebsiella pneumoniae Pathogen PF00753 8.1 IC50 BindingDB