Molecule Details
InChIKeyWYBRFXSHAXWYIZ-UHFFFAOYSA-N
Compound Name4-(2-fluorophenyl)-3,7,7-trimethyl-4,6,8,9-tetrahydro-2H-pyrazolo[3,4-b]quinolin-5-one
Canonical SMILESCc1n[nH]c2c1C(c1ccccc1F)C1=C(CC(C)(C)CC1=O)N2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.98
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49840 GSK3A Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
P49841 GSK3B Homo sapiens Human PF00069 6.7 Kd ChEMBL;BindingDB
P48730 CSNK1D Homo sapiens Human PF00069 6.5 Ki ChEMBL