Molecule Details
InChIKeyWXRGFPHDRFQODR-ICLZECGLSA-N
Canonical SMILESCC(C)N(CCCNC(=O)Nc1ccc(C(C)(C)C)cc1)C[C@H]1O[C@@H](n2ccc3c(N)ncnc32)[C@H](O)[C@@H]1O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.85
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q8TEK3 DOT1L Homo sapiens Human PF08123 9.4 IC50 ChEMBL;BindingDB
O14744 PRMT5 Homo sapiens Human PF05185 PF17286 PF17285 6.3 IC50 ChEMBL