Molecule Details
InChIKeyWXMCOSHTOJTIFK-UHFFFAOYSA-N
Compound NameN-[2-[[5-chloro-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]amino]phenyl]prop-2-enamide
Canonical SMILESC=CC(=O)Nc1ccccc1Nc1nc(Nc2ccnn2C)ncc1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.24
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28482 MAPK1 Homo sapiens Human PF00069 7.9 IC50 ChEMBL;BindingDB
P27361 MAPK3 Homo sapiens Human PF00069 6.9 IC50 ChEMBL
Q02750 MAP2K1 Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB