Molecule Details
InChIKeyWXGFWVAZGIOWBV-UHFFFAOYSA-N
Compound Name3-methylbutyl N-[2-[3-fluoro-4-[[6-(morpholine-4-carbonylamino)-4-oxo-2-propylquinazolin-3-yl]methyl]phenyl]phenyl]sulfonylcarbamate
Canonical SMILESCCCc1nc2ccc(NC(=O)N3CCOCC3)cc2c(=O)n1Cc1ccc(-c2ccccc2S(=O)(=O)NC(=O)OCCC(C)C)cc1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.82
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30556 AGTR1 Homo sapiens Human PF00001 9.2 IC50 ChEMBL;BindingDB
P50052 AGTR2 Homo sapiens Human PF00001 8.5 IC50 ChEMBL;BindingDB