Molecule Details
InChIKeyWXGCJNLWHYWDFU-KRWDZBQOSA-N
Compound Name2''-Cyclohexylamino-6-((S)-pyrrolidin-3-ylamino)[2,4'']bipyridinyl-4-carboxylic Acid Amide
Canonical SMILESNC(=O)c1cc(N[C@H]2CCNC2)nc(-c2ccnc(NC3CCCCC3)c2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.57
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15139 PRKD1 Homo sapiens Human PF00130 PF00169 PF00069 PF25525 7.2 IC50 ChEMBL;BindingDB
Q13563 PKD2 Homo sapiens Human PF18109 PF08016 PF20519 6.3 IC50 BindingDB
Q9BZL6 PRKD2 Homo sapiens Human PF00130 PF00169 PF00069 PF25525 6.3 IC50 ChEMBL