Molecule Details
InChIKeyWXCYFVSQEDOICZ-UHFFFAOYSA-N
Compound NameN-(1-(pyridin-4-yl)ethyl)-5-(2,2,2-trifluoroacetyl)thiophene-2-carboxamide
Canonical SMILESCC(NC(=O)c1ccc(C(=O)C(F)(F)F)s1)c1ccncc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.59
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q02161 RHD Homo sapiens Human PF00909 6.6 pIC50 TTD_MultiTarget
Q13547 HDAC1 Homo sapiens Human PF00850 6.6 pIC50 TTD_MultiTarget
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 6.6 IC50 ChEMBL;BindingDB