Molecule Details
InChIKeyWVWKMLRXXWPJFD-YWKITWBDSA-N
Canonical SMILES[C]N([C])[C]1[C]=[C]C2=C(c3ccc(C([O])=O)cc3C(=O)[N][C@H]([C][C][C][C][N])C(=O)[N]C([N])=N[C][C][C][C@@H]([N]C(=O)[C@@H]([C][C][C]N=C([N])[N])[N]C(=O)[C@@H]([C][C][C]N=C([N])[N])[N]C(=O)[C@@H]([C][C][C]N=C([N])[N])[N]C(=O)[C@@H]([C][C][C]N=C([N])[N])[N]C(=O)[C@@H]([C][C][C]N=C([N])[N])[N]C(=O)[C][C][C][C][C][N][C][C][N]S(=O)(=O)c3cccc4cnccc34)C([N])=O)c3ccc(N([C])[C])cc3OC2=[C]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.24
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13976 PRKG1 Homo sapiens Human PF00027 PF16808 PF00069 8.5 Kd BindingDB
O75582 RPS6KA5 Homo sapiens Human PF00069 PF00433 8.3 Kd BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 8.0 Kd BindingDB