Molecule Details
InChIKeyWVAWTXJGGXPRFT-CDHQVMDDSA-N
Canonical SMILESO=C(O)c1ccc(NC(=O)[C@H](C[C@H]2CC[C@H](O)CC2)c2ccc(-c3c(OC(F)F)ccc(Cl)c3F)c[n+]2[O-])cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.88
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P03951 F11 Homo sapiens Human PF00024 PF00089 9.8 IC50 ChEMBL;BindingDB
P03952 KLKB1 Homo sapiens Human PF00024 PF00089 7.9 IC50 ChEMBL;BindingDB