Molecule Details
InChIKeyWUSIUKLVFNJEHL-ZCYQVOJMSA-N
Compound Name(3R,3aR)-3-[[4-(naphthalen-2-ylmethyl)piperazin-1-yl]methyl]-3,3a,4,5-tetrahydro-[1,2]oxazolo[4,3-c]quinoline
Canonical SMILESc1ccc2c(c1)NC[C@@H]1C2=NO[C@H]1CN1CCN(Cc2ccc3ccccc3c2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 9.3 Ki ChEMBL;BindingDB
P08913 ADRA2A Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB
P18825 ADRA2C Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB