Molecule Details
InChIKeyWUKDUCCXRVBEIK-ZVHZXABRSA-N
Compound Name(5E)-4-methyl-5-[4-[(2,3,4,5,6-pentafluorophenyl)sulfonylamino]phenyl]sulfonylimino-1,3,4-thiadiazole-2-sulfonamide
Canonical SMILESCn1nc(S(N)(=O)=O)s/c1=N/S(=O)(=O)c1ccc(NS(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.44
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 8.8 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.8 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 7.7 Ki ChEMBL;BindingDB