Molecule Details
InChIKeyWUANZGDSZKKACG-KCWPFWIISA-N
Compound Name4-[2-[(2S,4R)-6-carbamimidoyl-4-phenyl-1,2,3,4-tetrahydroquinolin-2-yl]phenyl]benzene-1,3-dicarboxylic acid
Canonical SMILESN=C(N)c1ccc2c(c1)[C@@H](c1ccccc1)C[C@@H](c1ccccc1-c1ccc(C(=O)O)cc1C(=O)O)N2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.87
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P03951 F11 Homo sapiens Human PF00024 PF00089 8.1 Ki ChEMBL;BindingDB
P08709 F7 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 6.5 Ki ChEMBL
P00742 F10 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 6.0 Ki ChEMBL;BindingDB