Molecule Details
InChIKeyWTSMHXPVVATNPR-UHFFFAOYSA-N
Compound NameN-[2-methoxy-5-[[1-[2-(2-methylquinolin-5-yl)oxyethyl]piperidin-4-yl]methyl]phenyl]methanesulfonamide
Canonical SMILESCOc1ccc(CC2CCN(CCOc3cccc4nc(C)ccc34)CC2)cc1NS(C)(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.5
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28221 HTR1D Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB