Molecule Details
InChIKeyWTRQXHALVSEXHZ-UHFFFAOYSA-N
Compound NameN1-(4-(2-chlorophenyl)-6-(2-(isopropylamino)thiazol-5-yl)pyrimidin-2-yl)-N2,N2-dimethylethane-1,2-diamine
Canonical SMILESCC(C)Nc1ncc(-c2cc(-c3ccccc3Cl)nc(NCCN(C)C)n2)s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.41
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P53671 LIMK2 Homo sapiens Human PF00412 PF00595 PF07714 8.5 IC50 ChEMBL;BindingDB
P53667 LIMK1 Homo sapiens Human PF00412 PF00595 PF07714 8.4 IC50 ChEMBL;BindingDB
Q16539 MAPK14 Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB