Molecule Details
InChIKeyWTEGSNARHOVIJM-NUHJPDEHSA-N
Compound NameN2-((S)-1-(1H-benzo[d]iMidazol-5-yl)ethyl)-N4-(5-(2,2-difluorocyclopropyl)-1H-pyrazol-3-yl)pyriMidine-2,4-diaMine
Canonical SMILESC[C@H](Nc1nccc(Nc2cc(C3CC3(F)F)[nH]n2)n1)c1ccc2[nH]cnc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.89
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13153 PAK1 Homo sapiens Human PF00786 PF00069 7.5 IC50 ChEMBL;BindingDB
O75914 PAK3 Homo sapiens Human PF00786 PF00069 6.6 IC50 ChEMBL;BindingDB
Q13177 PAK2 Homo sapiens Human PF00786 PF00069 6.6 IC50 ChEMBL;BindingDB