Molecule Details
InChIKeyWTCGFNGKABLMFK-JDPFVKLISA-N
Compound NameH-2Nal-Cys(1)-3Pal-D-Trp-Lys-Ala-Cys(1)-2Nal-NH2
Canonical SMILESC[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2cccnc2)NC(=O)[C@@H](NC(=O)[C@@H](N)Cc2ccc3ccccc3c2)CSSC[C@@H](C(=O)N[C@@H](Cc2ccc3ccccc3c2)C(N)=O)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30874 SSTR2 Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB
P32745 SSTR3 Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB