Molecule Details
InChIKeyWTBNAFYSFOUZGF-UHFFFAOYSA-N
Compound Name4-(2,4-dimethyl-1,3-thiazol-5-yl)-N-(3-fluorophenyl)pyrimidin-2-amine
Canonical SMILESCc1nc(C)c(-c2ccnc(Nc3cccc(F)c3)n2)s1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.0
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.0 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 7.0 pIC50 TTD_MultiTarget