Molecule Details
InChIKeyWSQSTYRDZFLOBK-UCRWPKHMSA-N
Compound NameN-[3-[2-[2-[3-[[2-[2-[[(4R,9S,12S,15S,18S,21S,24R)-4-[(2-amino-2-oxoethyl)carbamoyl]-9,18-dibenzyl-15-(3-carbamimidamidopropyl)-21-[(1R)-1-hydroxyethyl]-6,8,11,14,17,20,23-heptaoxo-12-propan-2-yl-1,2-dithia-5,7,10,13,16,19,22-heptazacyclopentacos-24-yl]amino]-2-oxoethoxy]acetyl]amino]propoxy]ethoxy]ethoxy]propyl]-N'-[(2S,3R,4R,6R)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]-N'-methylbutanediamide
Canonical SMILESCO[C@@H]1[C@H](N(C)C(=O)CCC(=O)NCCCOCCOCCOCCCNC(=O)COCC(=O)N[C@H]2CSSC[C@@H](C(=O)NCC(N)=O)NC(=O)NC(=O)[C@H](Cc3ccccc3)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](Cc3ccccc3)NC(=O)[C@H]([C@@H](C)O)NC2=O)C[C@H]2O[C@]1(C)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.59
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P17612 PRKACA Homo sapiens Human PF00069 8.6 IC50 ChEMBL
P22612 PRKACG Homo sapiens Human PF00069 8.6 IC50 ChEMBL
P22694 PRKACB Homo sapiens Human PF00069 8.6 IC50 ChEMBL