Molecule Details
InChIKeyWSCBMCCISYODBR-XKZIYDEJSA-N
Compound Name1-[(3,4-difluorophenyl)methyl]-N-[4-[[(3Z)-3-(1H-imidazol-5-ylmethylidene)-2-oxo-1H-indol-5-yl]amino]-4-oxobutyl]-2-oxopyridine-3-carboxamide
Canonical SMILESO=C(CCCNC(=O)c1cccn(Cc2ccc(F)c(F)c2)c1=O)Nc1ccc2c(c1)/C(=C/c1cnc[nH]1)C(=O)N2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.48
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O15530 PDPK1 Homo sapiens Human PF14593 PF00069 6.6 IC50 ChEMBL;BindingDB
Q15118 PDK1 Homo sapiens Human PF10436 PF02518 6.6 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB