Molecule Details
InChIKeyWRYKLWBWSPEKIL-UHFFFAOYSA-N
Compound NameN-(2-amino-5-phenylphenyl)-8-cyclopropyl-7-piperazin-1-ylquinoline-3-carboxamide
Canonical SMILESNc1ccc(-c2ccccc2)cc1NC(=O)c1cnc2c(C3CC3)c(N3CCNCC3)ccc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13547 HDAC1 Homo sapiens Human PF00850 8.1 IC50 ChEMBL;BindingDB
Q92769 HDAC2 Homo sapiens Human PF00850 7.8 IC50 ChEMBL;BindingDB
O15379 HDAC3 Homo sapiens Human PF00850 6.8 IC50 ChEMBL;BindingDB