Molecule Details
InChIKeyWRLALEDDWSKGGQ-UHFFFAOYSA-N
Compound Name6-[2-[[2-hydroxy-3-(1H-indol-4-yloxy)propyl]amino]propoxy]-4H-1,4-benzoxazin-3-one
Canonical SMILESCC(COc1ccc2c(c1)NC(=O)CO2)NCC(O)COc1cccc2[nH]ccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.4
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P07550 ADRB2 Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 7.3 Ki ChEMBL;BindingDB